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Natural Science, Biology, 2024, 14, 67–75
DOI: 10.xxxx/example-doi Special Issue 1(2), 2022 186–1928

CONVENIENT APPROACH TO SYNTHESIS OF ALKALOID CERPEGIN DERIVATIVESv

Received N/A; revised N/A; accepted N/A
CC BY-NC 4.0 This work is licensed under Creative Commons Attribution–NonCommercial International License (CC BY-NC 4.0).

A convenient method for obtaining pyridine alkaloid cerpegin and its various new C-1 and N-5 derivatives in high yields has been developed. Starting enaminolactones, synthesized by means of various tertiary keto-alcohols, have been condensed with primary aliphatic, aromatic or heterocyclic amines for a pyridine cycle formation. Bromine derivatives of furo[3,4-c]pyridinenones are obtained as well.

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